Open main menu
Opium poppy (Papaver somniferum) flower

This is a list of opioids, opioid antagonists and inverse agonists.

Opium and poppy straw derivativesEdit

 
Seedhead of opium poppy with white latex

Crude opiate extracts whole opium productsEdit

Natural opiatesEdit

Opium alkaloidsEdit

Alkaloid salts mixturesEdit

Semisynthetics including Bentley compoundsEdit

Morphine familyEdit

3,6-diesters of morphineEdit

Codeine-dionine familyEdit

Morphinones and morpholsEdit

MorphidesEdit

Dihydrocodeine seriesEdit

Nitrogen morphine derivativesEdit

HydrazonesEdit

Structures
Hydrazones
  Oxymorphazone

Halogenated morphine derivativesEdit

Structures

Active opiate metabolitesEdit

MorphinansEdit

BenzomorphansEdit

4-PhenylpiperidinesEdit

Pethidines (meperidines)Edit

ProdinesEdit

KetobemidonesEdit

OthersEdit

Structures
Other phenylpiperidines
 Alvimopan   Loperamide   Picenadol

Open chain opioidsEdit

AmidonesEdit

MethadolsEdit

MoramidesEdit

ThiambutenesEdit

PhenalkoxamsEdit

AmpromidesEdit

Structures

OthersEdit

Structures
Other open chain opioids
 

Embutramide

 

IC-26

 

Isoaminile

 

Lefetamine

 

R-4066

AnilidopiperidinesEdit

Oripavine derivativesEdit

PhenazepanesEdit

PirinitramidesEdit

Structures
Pirinitramides
 

Bezitramide

 

Piritramide

BenzimidazolesEdit

IndolesEdit

Beta-Amino KetonesEdit

DiphenylmethylpiperazinesEdit

Opioid peptidesEdit

OthersEdit

Opioid antagonists and inverse agonistsEdit

Biased ligandsEdit

Receptor heteromer targeting ligandsEdit

Uncategorized opioidsEdit

Combination drug formulations containing opioidsEdit

See alsoEdit

ReferencesEdit

  1. ^ ChemIndex CAS Registry Number 3371-56-0
  2. ^ ChemIndex CAS Registry Number 509-56-8
  3. ^ ChemIndex CAS Registry Number 63715-94-6
  4. ^ NCBI PubChem SID 750205
  5. ^ chembase[permanent dead link] cbid_346222
  6. ^ Gomes I, Fujita W, Gupta A, Saldanha SA, Saldanha AS, Negri A, Pinello CE, Eberhart C, Roberts E, Filizola M, Hodder P, Devi LA (2013). "Identification of a μ-δ opioid receptor heteromer-biased agonist with antinociceptive activity". Proc. Natl. Acad. Sci. U.S.A. 110 (29): 12072–7. Bibcode:2013PNAS..11012072G. doi:10.1073/pnas.1222044110. PMC 3718106. PMID 23818586.
  7. ^ Yekkirala AS, Lunzer MM, McCurdy CR, Powers MD, Kalyuzhny AE, Roerig SC, Portoghese PS (2011). "N-naphthoyl-beta-naltrexamine (NNTA), a highly selective and potent activator of μ/kappa-opioid heteromers". Proc. Natl. Acad. Sci. U.S.A. 108 (12): 5098–103. Bibcode:2011PNAS..108.5098Y. doi:10.1073/pnas.1016277108. PMC 3064379. PMID 21385944.

External linksEdit

  • Carbonate derivatives of 14β-hydroxycodeine "viz., 14β-hydroxy-6-O-(methoxycarbonyl)codeine, 6-O-methoxycarbonyl-14β-(methoxycarbonyloxy)codeine, and 14β-acetoxy-6-O-methoxy-carbonylcodeine, potential substrates for ring C modification in morphinane (sic) alkaloids, were synthesized for the first time." Russian Chemical Bulletin. August 2008, Volume 57, Issue 8, pp 1773–1774. Date: 11 Aug 2009; I. V. Evsikova, S. K. Moiseev, P. V. Petrovskii, V. N. Kalinin. Published in Russian in Izvestiya Akademii Nauk. Seriya Khimicheskaya, No. 8, pp. 1739–1740