WIN 54,461 (6-Bromopravadoline) is a drug that acts as a potent and selective inverse agonist for the cannabinoid receptor CB2.[1]

WIN 54,461
Identifiers
  • [6-bromo-2-methyl-1-(2-morpholin-4-ylethyl)-1H-indol-3-yl](4-methoxyphenyl)methanone
PubChem CID
ChemSpider
Chemical and physical data
FormulaC23H25BrN2O3
Molar mass457.368 g·mol−1
3D model (JSmol)
  • Brc4ccc2c(n(c(c2C(=O)c1ccc(OC)cc1)C)CCN3CCOCC3)c4

See also edit

References edit

  1. ^ Howlett AC, Berglund B, Melvin LS (October 1995). "Cannabinoid Receptor Agonists and Antagonists". Current Pharmaceutical Design. 1 (3): 343–352. doi:10.2174/1381612801666220918164118. S2CID 252386978.